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Design and synthesis of endoperoxide antimalarial prodrug models

  • Paul M. O'Neill
  • , Paul A. Stocks
  • , Matthew D. Pugh
  • , Nuna C. Araujo
  • , Edward E. Korshin
  • , Jamie F. Bickley
  • , Steve Ward
  • , Patrick G. Bray
  • , Erica Pasini
  • , Jill Davies
  • , Edite Verissimo
  • , Mario D. Bachi
  • University of Liverpool
  • Weizmann Institute of Science
  • Liverpool School of Tropical Medicine

Research output: Contribution to journalArticlepeer-review

62 Citations (Scopus)
Original languageEnglish
Pages (from-to)4193-4197
Number of pages5
JournalAngewandte Chemie - International Edition
Volume43
Issue number32
DOIs
Publication statusPublished - 13 Aug 2004

Keywords

  • Antimalarial agents
  • Chalcones
  • Combination chemotherapy
  • Cysteine protease inhibitors
  • Endoperoxides

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